科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 耳草
英文名称: Auricled Hedyotis
拉丁名称: Hedyotis auricularia
使用部位: whole herb
功用: To clear heat and resolve toxin, cool blood and disperse swelling.
适用症: Common cold with fever, lung heat cough, swelling pain in throat, enteritis, dysentery, bleeding from hemorrhoids, flooding and spotting, poisonous snake bite, mastitis, swelling toxin of welling abscess and boil, eczema, knocks and falls.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
14259-45-1 车叶草苷 Asperuloside 84298
25368-11-0 车叶草苷酸 Asperulosidic acid 11968867
73706-32-8 - Auricularine 441990
83-46-5 β-谷甾醇 Beta-Sitosterol 222284
107-43-7 甜菜碱 Betaine 247
62-49-7 2-羟基-N,N,N-三甲基乙铵 Choline 305
14260-99-2 车叶草苷酸甲酯 Daphylloside 21602024
520-18-3 山柰素(山柰酚) Kaempferol 5280863
83-48-7 豆甾醇 Stigmasterol 5280794

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
APP AAA; ABETA; ABPP; AD1; APPI; CTFgamma; CVAP; PN-II; PN2; preA4 21q21.3 24107941
BACE1 ASP2; BACE; HSPC104 11q23.3 24107941
CHRNA7 CHRNA7-2; NACHRA7 15q13.3 31560162
NR1H2 LXR-b; LXRB; NER; NER-I; RIP15; UNR 19q13.33 24107776
NR1H3 LXR-a; LXRA; RLD-1 11p11.2 24107776
NR1H4 BAR; FXR; HRR-1; HRR1; PFIC5; RIP14 12q23.1 24107776

4. 相关疾病

疾病名称 疾病类型 参考文献
Aging phenotype 24932939
Alzheimer's Disease disease 31560162
Down Syndrome disease 24932939
Liver diseases group 24107776
Trisomy group 24932939