科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 橡皮木
英文名称: Common Alstonia
拉丁名称: Alstonia scholaris
使用部位: bark or leaf
功用: To clear heat and resolve toxin, relieve cough and dispel phlegm, stanch bleeding and disperse swelling.
适用症: Common cold with fever, lung heat cough asthma, pertussis, icterohepatitis, stomachache, vomiting and diarrhea, malaria, swollen welling abscess and sores, painful swelling from knocks and falls, bleeding due to external injury.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
5096-57-1 (-)-四氢小檗碱 (S)-Canadine 21171
650-69-1 - beta-Citraurin 9845703
20972-07-0 - Campesteryl Ferulate 15056832
88798-74-7 - Eckol 145937
486-70-4 羽扇豆宁 Lupinine 91461
138-55-6 苦番红花素;苦藏花素 Picrocrocin 130796
83-48-7 豆甾醇 Stigmasterol 5280794
6711-69-9 - Tubotaiwine 13783720
863-76-3 α-香树脂醇乙酸酯 α-Amyrin acetate 92842

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
APP AAA; ABETA; ABPP; AD1; APPI; CTFgamma; CVAP; PN-II; PN2; preA4 21q21.3 24107941
BACE1 ASP2; BACE; HSPC104 11q23.3 24107941
NR1H2 LXR-b; LXRB; NER; NER-I; RIP15; UNR 19q13.33 24107776
NR1H3 LXR-a; LXRA; RLD-1 11p11.2 24107776
NR1H4 BAR; FXR; HRR-1; HRR1; PFIC5; RIP14 12q23.1 24107776
TLR4 ARMD10; CD284; TLR-4; TOLL 9q33.1 24107776

4. 相关疾病

疾病名称 疾病类型 参考文献
Liver diseases group 24107776