科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 东北延胡索
英文名称: Amur Corydalis Equivalent plant: Corydalis repens
拉丁名称: Corydalis ambigua var. amurensis [Syn. Corydalis a
使用部位: tuber
功用: To quicken blood and dissipate stasis, rectify qi and relieve pain.
适用症: Pain in lumbus and knees, pain in heart and abdomen, dysmenorrhea, menstrual disorder, postpartum stasis stagnation abdominal pain, flooding and spotting, concretion and conglomeration, knocks and falls.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
24240-04-8 别隐品碱 Allocryptopine 98570
485-49-4 荷包牡丹碱 Bicuculline 10237
3486-66-6 黄连碱 Coptisine 72322
30045-16-0 脱氢紫堇碱 Dehydrocorydaline 34781
475-81-0 海罂粟碱 Glaucine 16754
3486-67-7 掌叶防已碱;巴马汀 Palmatine 19009
130-86-9 原阿片碱 Protopine 4970

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
BCL2 Bcl-2; PPP1R50 18q21.33 22033245
CASP1 ICE; IL1BC; P45 11q22.3 31336157
CDK1 CDC2; CDC28A; P34CDC2 10q21.2 22033245
GRIA2 GLUR2; GLURB; GluA2; GluR-K2; HBGR2; gluR-2; gluR-B 4q32.1 21414928
MCL1 BCL2L3; EAT; MCL1-ES; MCL1L; MCL1S; Mcl-1; TM; bcl2-L-3; mcl1/EAT 1q21.2 22033245
NLRP3 AGTAVPRL; AII; AVP; C1orf7; CIAS1; CLR1.1; DFNA34; FCAS; FCAS1; FCU; KEFH; MWS; NALP3; PYPAF1 1q44 31336157

4. 相关疾病

疾病名称 疾病类型 参考文献
Neoplasms, Hormone-Dependent phenotype 22033245
Prostatic Neoplasms group 22033245