科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 沉香
英文名称: Oily wood of Agalloch Eaglewood
拉丁名称: Lignum Aquilariae Resitum
使用部位: resinous wood
功用: To promote the flow of qi and relieve pain, to arrest vomiting by warming the stomach, and to relieve asthma.
适用症: Cold pain in stomach duct and abdomen, qi counterflow with asthma, stomach cold with retching counterflow, vacuity cold in lumbus and knees, vacuity constipation, qi strangury.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
13877-91-3 罗勒烯 - 5281553
2243-33-6 - (+)-alpha-Phellandrene 443160
489-39-4 (+)-Aromadendrene (+)-Aromadendrene 11095734
5794-03-6 - (+)-Camphene 92221
7785-26-4 (1S)-(-)-α-蒎烯 (-)-alpha-Pinene 440968
577-27-5 - (1aR,4R,4aS,7R,7aS,7bS)-1,1,4,7-tetramethyl-2,3,4a,5,6,7,7a,7b-octahydro-1aH-cyclopropa[e]azulen-4-ol 92812
52483-01-9 - (2S)-2-(2,4-dihydroxyphenyl)-5,7-dihydroxy-8-[(2R)-5-hydroxy-5-methyl-2-prop-1-en-2-ylhexyl]-2,3-dihydrochromen-4-one 44563159
629-96-9 1-二十醇 1-Eicosanol 12404
4176-97-0 14-去氧穿心莲内酯 14-Deoxyandrographolide 11624161
96-76-4 2,4-二叔丁基酚 2,4-Di-tert-butylphenol 7311

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ADAMTS4 ADAMTS-2; ADAMTS-4; ADMP-1 1q23.3 28237856
ADIPOQ ACDC; ACRP30; ADIPQTL1; ADPN; APM-1; APM1; GBP28 3q27.3 23623334
AGTR1 AG2S; AGTR1B; AT1; AT1AR; AT1B; AT1BR; AT1R; AT2R1; HAT1R 3q24 23992296
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 25260383
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24157255
ALPL AP-TNAP; APTNAP; HOPS; TNALP; TNAP; TNSALP 1p36.12 25832436
ALPP ALP; ALPI; IAP; PALP; PLAP; PLAP-1 2q37.1 25832436
ASRGL1 ALP; ALP1; CRASH 11q12.3 25832436
ATHS ALP 19p13.3-p13.2 25832436
ATRNL1 ALP; bA338L11.1; bA454H24.1 10q25.3 25832436

4. 相关疾病