科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 杜仲
英文名称: Eucommia bark
拉丁名称: Cortex Eucommiae
使用部位: bark
功用: To tonify the liver and the kidney, to strengthen the tendons and bones, and to prevent miscarrige.
适用症: Hypertension, kidney vacuity lumbago, weakness in sinews and bones, stirring fetus in pregnancy.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
506-30-9 花生酸 - 10467
35323-91-2 - (+)-Epicatechin 182232
29106-36-3 松脂素二甲醚 (+)-Eudesmin 73117
29106-36-3 松脂素二甲醚 (+)-Eudesmin 73117
38916-91-5 erythro-Guaiacylglycerol (1R,2S)-1-(4-hydroxy-3-methoxyphenyl)propane-1,2,3-triol 51382654
119677-21-3 (3R)-3-Hydroxy-D-proline (2R,3R)-3-hydroxypyrrolidine-2-carboxylic acid 10725382
118492-86-7 顺式-3-羟基-D-脯氨酸 (2R,3S)-3-hydroxypyrrolidine-2-carboxylic acid 11137200
69251-96-3 (+)松脂素-β-D-吡喃葡萄糖苷 (2S,3R,4S,5S,6R)-2-[4-[(3S,3aR,6S,6aR)-3-(4-hydroxy-3-methoxyphenyl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-6-yl]-2-methoxyphenoxy]-6-(hydroxymethyl)oxane-3,4,5-triol 486614
105279-10-5 柑属苷B (2S,3R,4S,5S,6R)-2-[4-[1,3-Dihydroxy-2-[4-[(E)-3-hydroxyprop-1-enyl]-2,6-dimethoxyphenoxy]propyl]-2-methoxyphenoxy]-6-(hydroxymethyl)oxane-3,4,5-triol 11972318
6532-76-9 - (3R)-3-hydroxy-L-aspartic acid 14463

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 21445586
ABCC3 ABC31; EST90757; MLP2; MOAT-D; MRP3; cMOAT2 17q21.33 23847194
ABCG2 ABC15; ABCP; BCRP; BCRP1; BMDP; CD338; CDw338; EST157481; GOUT1; MRX; MXR; MXR-1; MXR1; UAQTL1 4q22.1 21625222
ACTA2 ACTSA 10q23.31 22302193
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 25950476
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 20840540
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21168456
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21708244
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24000005
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27472952

4. 相关疾病