科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 半枝莲
英文名称: all - grass of Barbed Skullcap
拉丁名称: Herba Scutellariae barbatae
使用部位: whole herb
功用: To remove toxic heat, and to cause diuresis.
适用症: Heat toxin swollen welling abscess, throat pain, pulmonary welling abscess, intestinal welling abscess, scrofula, poisonous snake bite, knocks and falls, blood ejection, spontaneous external bleeding, blood strangury, edema, ascites, carcinoma.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
499-94-5 - (+)-p-Menth-1-ene 11815433
464-48-2 - (-)-Camphor 444294
2181-76-2 - (2S)-4-[2-[(2S)-2-carboxy-5,6-dihydroxy-2,3-dihydroindol-1-yl]ethenyl]-2,3-dihydropyridine-2,6-dicarboxylic acid 137218006
3687-48-7 - (3R)-oct-1-en-3-ol 6992244
7362-39-2 p-Coumaric acid ethyl ester (E)-Ethyl 3-(4-hydroxyphenyl)acrylate 676946
111-27-3 正己醇 1-Hexanol 8103
100079-39-8 2',4'-Dihydroxy-2,3',6'-trimethoxychalcone 2',4'-Dihydroxy-2,3',6'-trimethoxychalcone 21636239
496-16-2 - 2,3-Dihydrobenzofuran 10329
6728-26-3 反式-2-己烯醛 2-Hexenal 5281168
17241-40-6 2-羟基-3-甲基蒽醌 2-Hydroxy-3-methylanthraquinone 10889963

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
ADAMTS4 ADAMTS-2; ADAMTS-4; ADMP-1 1q23.3 28237856
ADIPOQ ACDC; ACRP30; ADIPQTL1; ADPN; APM-1; APM1; GBP28 3q27.3 23623334
AGT ANHU; SERPINA8; hFLT1 1q42.2 20942814
AHR RP85; bHLHe76 7p21.1 30166541
AHR RP85; bHLHe76 7p21.1 30831189
AHSA1 AHA1; C14orf3; hAha1; p38 14q24.3 20942814

4. 相关疾病