科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 毛冬青
英文名称: Pubescent Holly Equivalent plant: Ilex pubescens v
拉丁名称: Ilex pubescens
使用部位: root
功用: To clear heat and resolve toxin, quicken blood and free network vessels.
适用症: Angina pectoris, acute myocardial infarction, cerebral thrombosis, thrombophlebitis, thromboangiitis obliterans (Buerger’s disease), central retinitis, central angiospastic retinitis, wind-heat common cold, lung heat cough asthma, sore pharynx, nipple moth, gum swelling and pain, chest impediment and heart pain, wind stroke with hemiplegia, erysipelas, burns and scalds, welling abscess and flat abscess.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
645-08-9 异香草酸 3-Hydroxy-4-methoxybenzoic acid 12575
464-92-6 积雪草酸 Asiatic Acid 119034
85344-31-6 - Ilexolide A 441931
530-57-4 丁香酸 Syringic acid 10742
545-46-0 乌发醇 Uvaol 92802

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24486195
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21168456
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21708244
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24000005
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27472952
BAX BCL2L4 19q13.33 29228978
BBC3 JFY-1; JFY1; PUMA 19q13.32 24389342
BCL2 Bcl-2; PPP1R50 18q21.33 22832932
BCL2 Bcl-2; PPP1R50 18q21.33 27472952
BCL2L1 BCL-XL/S; BCL2L; BCLX; Bcl-X; PPP1R52 20q11.21 29228978

4. 相关疾病