科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 蔓荆子
英文名称: Shrub Chastetree Fruit
拉丁名称: Fructus Viticis
使用部位: seed
功用: To dispel wind-heat from the head and eyes.
适用症: Externally contracted wind-heat, dizziness and headache, migraine, gum swelling and pain, red eyes with gall, delacrimation, wind-damp impediment pain, hypertonicity of limbs.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
99-83-2 水芹烯 - 7460
483-76-1 (+)-DELTA-CADINENE - 441005
7785-70-8 (1R)-(+)-alpha-蒎烯 (+)-alpha-Pinene 82227
7785-53-7 - (+)-alpha-Terpineol 442501
7785-53-7 - (+)-alpha-Terpineol 442501
489-39-4 (+)-Aromadendrene (+)-Aromadendrene 11095734
19902-08-0 - (+)-beta-Pinene 10290825
5794-03-6 - (+)-Camphene 92221
2438-10-0 (+)-萜品-4-醇 (+)-Terpinen-4-ol 2724161
20296-50-8 - (-)-3-Carene 442461

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 30813295
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 25047426
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 20840540
APOE AD2; APO-E; ApoE4; LDLCQ5; LPG 19q13.32 31036637
APP AAA; ABETA; ABPP; AD1; APPI; CTFgamma; CVAP; PN-II; PN2; preA4 21q21.3 24107941
AURKA AIK; ARK1; AURA; BTAK; PPP1R47; STK15; STK6; STK7 20q13.2 25047426

4. 相关疾病