科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 化橘红
英文名称: Pummelo Peel
拉丁名称: Exocarpium Citri grandis
使用部位: -
功用: To dispel cold, eliminate damp and phlegm, and arrest emesis or nausea.
适用症: Treatment of cough, itching of the throat and profuse expectoration in colds, nausea, vomiting and epigastric distension caused by improper diet or excessive drinking.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
1460-97-5 - (-)-gamma-Cadinene 92313
480-41-1 - (2R)-5,7-dihydroxy-2-(4-hydroxyphenyl)-2,3-dihydro-4H-chromen-4-one 667495
6601-66-7 6-去甲氧基桔皮素 6-Demethoxytangeretin 629964
481-72-1 芦荟大黄素 Aloe emodin 10207
104-46-1 反式茴香脑 Anethole 637563
520-36-5 芹菜素 Apigenin 5280443
5631-70-9 4',5,7-三甲氧基黄酮 Apigenin trimethyl ether 79730
67979-25-3 橙黄决明素 Aurantio-obtusin 155011
67979-25-3 橙黄决明素 Aurantio-obtusin 155011
495-02-3 橙皮油素 Auraptene 1550607

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB1 ABC20; CD243; CLCS; GP170; MDR1; P-GP; PGY1 7q21.12 27058921
ABCB1 ABC20; CD243; CLCS; GP170; MDR1; P-GP; PGY1 7q21.12 28958806
ABCC1 ABC29; ABCC; GS-X; MRP; MRP1 16p13.11 28958806
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 28958806
AGT ANHU; SERPINA8; hFLT1 1q42.2 21844078
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21871133
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24157255
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27710830
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24125861
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24359639

4. 相关疾病