科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 厚朴
英文名称: Officinal Magnolia Equivalent plant: Magnolia bilo
拉丁名称: Magnolia officinalis
使用部位: bark
功用: To dry damp and disperse phlegm, precipitate qi and eliminate fullness, lower blood pressure.
适用症: Amebic dysentery, vomiting and diarrhea, food accumulation and qi stagnation, abdominal distention and constipation, phlegm-rheum cough asthma.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
495-61-4 (-)-β-bisabolene - 10104370
7785-70-8 (1R)-(+)-alpha-蒎烯 (+)-alpha-Pinene 82227
7785-53-7 - (+)-alpha-Terpineol 442501
51685-40-6 - (+)-Linalyl acetate 6999980
26871-46-5 Isomahanimbine (+)-Mahanimbicine 4072580
26871-46-5 Isomahanimbine (+)-Mahanimbicine 4072580
92829-72-6 Magnaldehyde B (E)-3-[4-hydroxy-3-(2-hydroxy-5-prop-2-enylphenyl)phenyl]prop-2-enal 5320888
115-71-9 - (Z)-5-[(1S,3R)-2,3-dimethyl-3-tricyclo[2.2.1.02,6]heptanyl]-2-methylpent-2-en-1-ol 24832102
470-67-7 1,4-桉叶素 1,4-Cineole 10106
20601-85-8 四氢厚朴酚 2-(2-Hydroxy-5-propylphenyl)-4-propylphenol 5321851

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ADAMTS4 ADAMTS-2; ADAMTS-4; ADMP-1 1q23.3 29649568
ADAMTS5 ADAM-TS 11; ADAM-TS 5; ADAM-TS5; ADAMTS-11; ADAMTS-5; ADAMTS11; ADMP-2 21q21.3 29649568
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 26454217
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27940017
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 30587839
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21757288
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 31905887
ALDH3A1 ALDH3; ALDHIII 17p11.2 29794221
BAX BCL2L4 19q13.33 22259050
BAX BCL2L4 19q13.33 29649568

4. 相关疾病

疾病名称 疾病类型 参考文献
Acute Lung Injury disease 21279327
Body mass index phenotype 26249791
Brain Edema phenotype 30597199
Brain Ischemia disease 30597199
Brain Neoplasms group 22259050
Cardiomegaly phenotype 25871545
Cerebral Hemorrhage phenotype 30597199
Endotoxemia phenotype 21279327
Fibrosis phenotype 21265825
Glioblastoma disease 30587839