科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 骨碎补
英文名称: rhizome of Heartleaf Dryria
拉丁名称: Rhizoma Dryriae
使用部位: rhizome
功用: To replenish the kidney, to strengthen the bones, to promote the healing of fracture, and to relieve pain.
适用症: Kidney vacuity lumbago, tinnitus and deafness, tooth mobilizing, wrenching and contusion from knocks and falls, sinew and bone wound, alopecia areata, white patch wind.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
24808-04-6 (-)-表阿夫儿茶精 (-)-Epiafzelechin 443639
480-41-1 - (2R)-5,7-dihydroxy-2-(4-hydroxyphenyl)-2,3-dihydro-4H-chromen-4-one 667495
69251-96-3 (+)松脂素-β-D-吡喃葡萄糖苷 (2S,3R,4S,5S,6R)-2-[4-[(3S,3aR,6S,6aR)-3-(4-hydroxy-3-methoxyphenyl)-1,3,3a,4,6,6a-hexahydrofuro[3,4-c]furan-6-yl]-2-methoxyphenoxy]-6-(hydroxymethyl)oxane-3,4,5-triol 486614
6638-05-7 2,6-Dimethoxy-4-Methylphenol 2,6-Dimethoxy-4-methylphenol 240925
91-10-1 2,6-二甲氧基苯酚 2,6-Dimethoxyphenol 7041
99282-79-8 2-(CARBOXYMETHYL-AMINO)-4-CHLORO-BENZOIC ACID 2-((Carboxymethyl)amino)-4-chlorobenzoic acid 11107141
67-47-0 5-羟甲基糠醛 5-Hydroxymethylfurfural 237332
67-47-0 5-羟甲基糠醛 5-Hydroxymethylfurfural 237332
2545-00-8 阿夫儿茶精 Afzelechin 442154
482-39-3 阿福豆苷 Afzelin 5316673

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 22607709
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 25047426
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27710830
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 20840540
APP AAA; ABETA; ABPP; AD1; APPI; CTFgamma; CVAP; PN-II; PN2; preA4 21q21.3 24107941
AURKA AIK; ARK1; AURA; BTAK; PPP1R47; STK15; STK6; STK7 20q13.2 25047426

4. 相关疾病