科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 盾叶薯蓣
英文名称: Peltate Ya m
拉丁名称: Dioscorea zingiberensis
使用部位: rhizome
功用: To clear lung and relieve cough, disinhibit damp and free strangury, free network vessels and relieve pain, resolve toxin and disperse swelling.
适用症: Lung heat cough, damp-heat strangury pain, wind-damp lumbago, swollen welling abscess and malign sore, sprain from knocks and falls, bee sting, insect bites.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
549-08-6 - (4aR)-3,4,4a,5,18,19-Hexahydro-9,21,22,26-tetramethoxy-4-methyl-2H-1,24:12,15-dietheno-6,10-metheno-16H-pyrido[2',3':17,18][1,10]dioxacycloeicosino[2,3,4-ij]isoquinoline 5317122
105454-04-4 7-表紫杉醇 7-epi-Taxol 184492
530-53-0 脱氧鸭嘴花碱酮 Deoxyvasicinone 68261
19083-00-2 纤细薯蓣皂苷 Gracillin 159861
87-52-5 芦竹碱 Gramine 6890

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
MAPK1 ERK; ERK-2; ERK2; ERT1; MAPK2; P42MAPK; PRKM1; PRKM2; p38; p40; p41; p41mapk; p42-MAPK 22q11.22 22461009
MAPK14 CSBP; CSBP1; CSBP2; CSPB1; EXIP; Mxi2; PRKM14; PRKM15; RK; SAPK2A; p38; p38ALPHA 6p21.31 21195543
MAPK3 ERK-1; ERK1; ERT2; HS44KDAP; HUMKER1A; P44ERK1; P44MAPK; PRKM3; p44-ERK1; p44-MAPK 16p11.2 22461009
NDUFA5 B13; CI-13KD-B; CI-13kB; NUFM; UQOR13 7q31.32 31649278
PDCD1 CD279; PD-1; PD1; SLEB2; hPD-1; hPD-l; hSLE1 2q37.3 30305604
PTGS2 COX-2; COX2; GRIPGHS; PGG/HS; PGHS-2; PHS-2; hCox-2 1q31.1 21195543
RPL17 L17; PD-1; RPL23 18q21.1 30305604
RPL17-C18orf32 PD-1; RPL17 18q21.1 30305604
SDHB CWS2; IP; PGL4; SDH; SDH1; SDH2; SDHIP 1p36.13 31649278
TNFRSF10B CD262; DR5; KILLER; KILLER/DR5; TRAIL-R2; TRAILR2; TRICK2; TRICK2A; TRICK2B; TRICKB; ZTNFR9 8p21.3 21195543

4. 相关疾病

疾病名称 疾病类型 参考文献
melanoma disease 30305604