科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 臭梧桐
英文名称: Glorybower leaf, Clerodendron leaf
拉丁名称: Folium Clerodentri trichotomi
使用部位: leaf
功用: To dispel wind and dampness
适用症: Hypertension, malaria, wind-damp impediment, numbness in limbs, hemiplegia, migraine, dysentery, hemorrhoids, welling abscess and flat abscess, scab sore.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
112-30-1 癸醇 1-Decanol 8174
19670-51-0 1-棕榈酸单甘油酯 2,3-Dihydroxypropyl hexadecanoate 14900
67-47-0 5-羟甲基糠醛 5-Hydroxymethylfurfural 237332
83-46-5 β-谷甾醇 Beta-Sitosterol 222284
105471-98-5 木通苯乙醇苷B Calceolarioside B 5273567
105471-98-5 木通苯乙醇苷B Calceolarioside B 5273567
35481-70-0 - Clerodendrin A 442013
10597-60-1 羟基酪醇 Hydroxytyrosol 82755
41546-34-3 D-手性肌醇 Inositol 892
61303-13-7 异麦角甾苷;异类叶升麻苷 Isoacteoside 6476333

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
ABCB11 ABC16; BRIC2; BSEP; PFIC-2; PFIC2; PGY4; SPGP 2q31.1 24107776
ABCC2 ABC30; CMOAT; DJS; MRP2; cMRP 10q24.2 24107776
ABCG5 STSL; STSL2 2p21 24107776
ABCG8 GBD4; STSL; STSL1 2p21 24107776
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24486741
APP AAA; ABETA; ABPP; AD1; APPI; CTFgamma; CVAP; PN-II; PN2; preA4 21q21.3 24107941
BACE1 ASP2; BACE; HSPC104 11q23.3 24107941
CRMP1 CRMP-1; DPYSL1; DRP-1; DRP1; ULIP-3 4p16.2 24316371
MAP3K14 FTDCR1B; HS; HSNIK; NIK 17q21.31 29505920
MGLL HU-K5; HUK5; MAGL; MGL 3q21.3 22646533

4. 相关疾病

疾病名称 疾病类型 参考文献
Hyperglycemia disease 24316371
Hyperlipidemia disease 24316371
Insulin Resistance phenotype 24316371
Liver diseases group 24107776
Liver neoplasms group 24486741
Melanoma, Experimental disease 29505920
Muscular Atrophy phenotype 24418157
Obesity disease 27940206
Obesity disease 24316371
Pain phenotype 22646533