科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 臭山羊
英文名称: Japanese Orixa
拉丁名称: Orixa japonica
使用部位: root
功用: To clear heat and resolve exterior, move qi and relieve pain, dispel wind and disinhibit damp.
适用症: Wind-heat common cold, cough, throat pain, toothache, stomachache, pain in joints due to rheumatalgia, dysentery, innominate toxin swelling.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
101330-69-2 3'-O-甲基山药素III 3'-O-Methylbatatasin III 442711
484-20-8 佛手柑内酯 Bergapten 2355
99-49-0 Carvone natural Carvone, (+/-)- 7439
1845-59-6 - Cyclohexanol, 2-methyl-5-(1-methylethyl)-, (1alpha,2beta,5alpha)- 6432473
5532-41-2 (8β,13β,14α,17β,18α,21β)-D:C-Friedo-B':A'-neogammacer-9(11)-en-3β-ol Isoarborinol 12305182
30426-61-0 - Japonine 442915
484-08-2 香草木宁 Kokusaginine 10227
68705-66-8 - Kolaflavanone 155169
50333-13-6 N-甲基芸香碱 N-Methylflindersine 72819
517-99-7 - Norpluviine 12313583

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
BAK1 BAK; BAK-LIKE; BCL2L7; CDN1 6p21.31 24680709
BAX BCL2L4 19q13.33 24680709
CYP3A4 CP33; CP34; CYP3A; CYP3A3; CYPIIIA3; CYPIIIA4; HLP; NF-25; P450C3; P450PCN1 7q22.1 29945292
IL10 CSIF; GVHDS; IL-10; IL10A; TGIF 1q32.1 27185659
MCL1 BCL2L3; EAT; MCL1-ES; MCL1L; MCL1S; Mcl-1; TM; bcl2-L-3; mcl1/EAT 1q21.2 24680709
NFKB1 CVID12; EBP-1; KBF1; NF-kB; NF-kB1; NF-kappa-B1; NF-kappaB; NF-kappabeta; NFKB-p105; NFKB-p50; NFkappaB 4q24 29945292
NR1I2 BXR; ONR1; PAR; PAR1; PAR2; PARq; PRR; PXR; SAR; SXR 3q13.33 29945292

4. 相关疾病

疾病名称 疾病类型 参考文献
Asthma disease 27185659
Bronchial Hyperreactivity disease 27185659
Colitis disease 29945292
Liver neoplasms group 24680709