科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 白鲜皮
英文名称: Densefruit Pittany Root-bark Equivalent plant: Dic
拉丁名称: Dictamnus dasycarpus
使用部位: root cortex
功用: To clear heat and dry damp, dispel wind and relieve itch, resolve toxin.
适用症: Dermatitis, psoriasis, icterohepatitis, damp-heat sore and papules, profuse pus, yellow-water sore, damp ulceration on skin, itchy skin, damp-heat jaundice, damp-heat impediment.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
751-29-1 - (2E)-3-[(3aS,5aR,6R,7R,9aR,9bR,10aS)-3-(Furan-3-yl)-7-(2-hydroxypropan-2-yl)-3a,6,9a-trimethyl-1,9-dioxododecahydronaphtho[2,1-c]oxireno[d]pyran-6-yl]prop-2-enoic acid 54611038
484-29-7 白鲜碱 Dictamnine 68085
28808-62-0 梣酮 Fraxinellone 124039
518-96-7 Isomaculosidine Furo(2,3-b)quinolin-4(9H)-one, 6,8-dimethoxy-9-methyl- 3083609
73793-68-7 Kihadanin B Kihadanin B 156766
1180-71-8 柠檬苦素(吴茱萸内酯) Limonin 179651
145-13-1 孕甾烯醇酮 Pregnenolone 8955
38695-41-9 前茵芋碱 Preskimmianine 12305721
83-95-4 茵芋碱(β-花椒碱) Skimmianine 6760
535-83-1 葫芦巴碱 Trigonelline 5570

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 25781227
CD274 B7-H; B7H1; PD-L1; PDCD1L1; PDCD1LG1; PDL1; hPD-L1 9p24.1 30103001
CLIP1 CLIP; CLIP-170; CLIP170; CYLN1; RSN 12q24.31 23955365
CNR1 CANN6; CB-R; CB1; CB1A; CB1K5; CB1R; CNR 6q15 24385629
CNR1 CANN6; CB-R; CB1; CB1A; CB1K5; CB1R; CNR 6q15 28220044
DCTN4 DYN4; P62 5q33.1 30339884
GABPA E4TF1-60; E4TF1A; NFT2; NRF2; NRF2A; RCH04A07 21q21.3 23108405
GABPA E4TF1-60; E4TF1A; NFT2; NRF2; NRF2A; RCH04A07 21q21.3 28012440
GABPA E4TF1-60; E4TF1A; NFT2; NRF2; NRF2A; RCH04A07 21q21.3 30339884
GPX4 GPx-4; GSHPx-4; MCSP; PHGPx; SMDS; snGPx; snPHGPx 19p13.3 30339884

4. 相关疾病