科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 徐长卿
英文名称: Paniculate Swallowwort Root
拉丁名称: Radix Cynchi Paniculati
使用部位: root
功用: To relieve rheumatic conditions, and to arrest pain and itching.
适用症: Rheumatic arthritis, toothache, lumbago, pain after operation, dysmenorrhea, mastitis, infection of skin, eczema, neurodermatitis, urticaria, infective dermatitis, zoster, wind-damp impediment pain, knocks and falls.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
32671-82-2 7-脱甲氧基娃儿藤碱 - 639288
14073-97-3 (-)-薄荷酮 (-)-Menthone 26447
17334-55-3 - (1aR,7R,7aR,7bS)-1,1,7,7a-tetramethyl-2,3,5,6,7,7b-hexahydro-1aH-cyclopropa[a]naphthalene 15560278
42075-32-1 (2R,4R)-(-)-2,4-戊二醇 (2R,4R)-(-)-Pentanediol 2723683
575-43-9 1,6-二甲基萘 1,6-Dimethylnaphthalene 11328
10139-84-1 2',4'-二羟基-3'-甲基苯乙酮 1-(2,4-Dihydroxy-3-methylphenyl)ethanone 592139
493-33-4 1-(4-羟基-2-甲氧基苯基)乙酮 1-(4-Hydroxy-2-methoxyphenyl)ethanone 529402
629-73-2 十六烯 1-Hexadecene 12395
90-12-0 - 1-Methylnaphthalene 7002
6869-50-7 - 14beta,17alpha-Pregn-5-en-20-one, 3beta,8,12beta,14-tetrahydroxy- 12311278

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 31406198
BAX BCL2L4 19q13.33 28456683
BCL2 Bcl-2; PPP1R50 18q21.33 28456683
CLDN1 CLD1; ILVASC; SEMP1 3q28 28456683
DGKD DGK-delta; DGKdelta; dgkd-2 2q37.1 28707095
IDO1 IDO; IDO-1; INDO 8p11.21 28456683
MLKL hMLKL 16q23.1 28456683
MTOR FRAP; FRAP1; FRAP2; RAFT1; RAPT1; SKS 1p36.22 31406198
MUC1 ADMCKD; ADMCKD1; CA 15-3; CD227; EMA; H23AG; KL-6; MAM6; MCD; MCKD; MCKD1; MUC-1; MUC-1/SEC; MUC-1/X; MUC1/ZD; PEM; PEMT; PUM 1q22 28456683
MUC2 MLP; MUC-2; SMUC 11p15.5 28456683

4. 相关疾病

疾病名称 疾病类型 参考文献
Colitis disease 28456683
Diabetes disease 28707095
Hyperglycemia disease 28707095