科华智慧(深圳)创新药物研发有限公司     西北农林科技大学深圳研究院    联合开发

1. 药材主信息

中文名称: 桔梗
英文名称: Platycodon Root
拉丁名称: Radix Platycodi
使用部位: root
功用: To relieve cought, to soothe sore throat, and to promote expectoration and discharge of pus.
适用症: Cough with profuse phlegm, swelling pain in throat, pulmonary welling abscess with hacking of pus and blood, fullness in chest and rib-side pain, dysentery, dribbling urinary block.
毒副作用: -

2. 相关成分

CAS号 中文名称 英文名称 参考文献
110979-06-1 - (2R)-1-(5-Methoxy-3,6-dioxocyclohexa-1,4-dien-1-yl)tridecan-2-yl acetate 46191017
480-41-1 - (2R)-5,7-dihydroxy-2-(4-hydroxyphenyl)-2,3-dihydro-4H-chromen-4-one 667495
66779-34-8 桔梗皂苷A 2''O-acetylplatycodin D 46173910
930-30-3 - 2-Cyclopenten-1-one 13588
66779-35-9 3’’-0-乙酰基-桔梗皂苷D 3''O-acetylplatycodin D 46173919
2454-31-1 - 3,4-Heptadiene 556860
29428-70-4 - 3beta-Hydroxy-28,13-ursanolide 131752032
1577-22-6 5-己烯酸 5-Hexenoic acid 15308
480-44-4 金合欢素;刺槐素 Acacetin 5280442
41547-82-4 腺苷 Adenosine 60961

3. 相关靶点

基因靶点 基因别名 靶点位置 参考文献
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27710830
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21168456
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 21708244
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 24000005
AKT1 AKT; CWS6; PKB; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA 14q32.33 27472952
BBC3 JFY-1; JFY1; PUMA 19q13.32 24389342
BCL2 Bcl-2; PPP1R50 18q21.33 22832932
BCL2 Bcl-2; PPP1R50 18q21.33 27472952
BCL2L1 BCL-XL/S; BCL2L; BCLX; Bcl-X; PPP1R52 20q11.21 22832932
BCL2L1 BCL-XL/S; BCL2L; BCLX; Bcl-X; PPP1R52 20q11.21 27472952

4. 相关疾病